Title : Structure-based discovery of novel 4,5,6-trisubstituted pyrimidines as potent covalent Bruton's tyrosine kinase inhibitors.

Pub. Date : 2016 Jul 1

PMID : 27210433






1 Functional Relationships(s)
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Protein Name
Organism
1 The preliminary structure-activity relationship was discussed and the primary amino group at the C-4 position of pyrimidine was crucial for maintaining BTK activity. pyrimidine Bruton tyrosine kinase Homo sapiens