Title : Kinetically Defined Mechanisms and Positions of Action of Two New Modulators of Glucocorticoid Receptor-regulated Gene Induction.

Pub. Date : 2016 Jan 1

PMID : 26504077






1 Functional Relationships(s)
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1 Consistent with its complicated biochemistry, BRD4 is shown to alter both the maximal activity (Amax) and the steroid concentration required for half-maximal induction (EC50) of GR-mediated gene expression by acting at a minimum of three different kinetically defined steps. Steroids nuclear receptor subfamily 3 group C member 1 Homo sapiens