Title : Modulation of P-glycoprotein at the Human Blood-Brain Barrier by Quinidine or Rifampin Treatment: A Positron Emission Tomography Imaging Study.

Pub. Date : 2015 Nov

PMID : 26354948






1 Functional Relationships(s)
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1 Furthermore, the magnitude of BBB P-gp inhibition by quinidine was successfully predicted by a combination of in vitro and macaque data, but not by rat data. Quinidine phosphoglycolate phosphatase Rattus norvegicus