Title : Identifying cytochrome p450 functional networks and their allosteric regulatory elements.

Pub. Date : 2013

PMID : 24312617






2 Functional Relationships(s)
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1 We investigated four CYP subfamilies (CYP1A, CYP2D, CYP2C, and CYP3A) that are involved in 90% of all metabolic drug transformations and identified four amino acid interaction networks associated with specific CYP functionalities, i.e., membrane binding, heme binding, catalytic activity, and dimerization. Heme cytochrome P450 family 4 subfamily F member 3 Homo sapiens
2 We investigated four CYP subfamilies (CYP1A, CYP2D, CYP2C, and CYP3A) that are involved in 90% of all metabolic drug transformations and identified four amino acid interaction networks associated with specific CYP functionalities, i.e., membrane binding, heme binding, catalytic activity, and dimerization. Heme cytochrome P450 family 4 subfamily F member 3 Homo sapiens