Title : Novel pyridazinone inhibitors for vascular adhesion protein-1 (VAP-1): old target-new inhibition mode.

Pub. Date : 2013 Dec 27

PMID : 24304424






3 Functional Relationships(s)
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1 Novel pyridazinone inhibitors for vascular adhesion protein-1 (VAP-1): old target-new inhibition mode. 2-phenyl-3(2H)-pyridazinone amine oxidase copper containing 3 Homo sapiens
2 Novel pyridazinone inhibitors for vascular adhesion protein-1 (VAP-1): old target-new inhibition mode. 2-phenyl-3(2H)-pyridazinone amine oxidase copper containing 3 Homo sapiens
3 Here we report the synthesis, inhibitory activity, and molecular binding mode of novel pyridazinone inhibitors, which show specificity for VAP-1 over monoamine and diamine oxidases. 2-phenyl-3(2H)-pyridazinone amine oxidase copper containing 3 Homo sapiens