Title : Potent P2Y1 urea antagonists bearing various cyclic amine scaffolds.

Pub. Date : 2013 Dec 15

PMID : 24269480






1 Functional Relationships(s)
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Protein Name
Organism
1 SAR optimization led to the identification of isoindoline 3c and piperidine 4a which showed good in vitro binding and functional activities, as well as improved aqueous solubility. piperidine sarcosine dehydrogenase Homo sapiens