Title : Cyclin-dependent kinase inhibitor dinaciclib interacts with the acetyl-lysine recognition site of bromodomains.

Pub. Date : 2013 Nov 15

PMID : 24007471






2 Functional Relationships(s)
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Protein Name
Organism
1 Remarkably, dinaciclib also interacted with the acetyl-lysine recognition site of the bromodomain testis-specific protein BRDT, a member of the BET family of bromodomains. dinaciclib bromodomain testis associated Homo sapiens
2 The binding mode of dinaciclib to BRDT at 2.0 A resolution suggests that general kinase inhibitors ("hinge binders") possess a previously unrecognized potential to act as protein-protein inhibitors of bromodomains. dinaciclib bromodomain testis associated Homo sapiens