Title : Pharmacological characterization of (3S)-3-(hydroxymethyl)-4-(5-methylpyridin-2-yl)-N-[6-(2,2,2-trifluoroethoxy)pyridin-3-yl]-3,4-dihydro-2H-benzo[b][1,4]oxazine-8-carboxamide (JTS-653), a novel transient receptor potential vanilloid 1 antagonist.

Pub. Date : 2012 Aug

PMID : 22588258






1 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 JTS-653 displaced [(3)H]resiniferatoxin binding to human and rat TRPV1. resiniferatoxin transient receptor potential cation channel, subfamily V, member 1 Rattus norvegicus