Title : Drug interaction of efavirenz and midazolam: efavirenz activates the CYP3A-mediated midazolam 1'-hydroxylation in vitro.

Pub. Date : 2012 Jun

PMID : 22415932






3 Functional Relationships(s)
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1 Drug interaction of efavirenz and midazolam: efavirenz activates the CYP3A-mediated midazolam 1"-hydroxylation in vitro. efavirenz cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 Drug interaction of efavirenz and midazolam: efavirenz activates the CYP3A-mediated midazolam 1"-hydroxylation in vitro. efavirenz cytochrome P450 family 3 subfamily A member 4 Homo sapiens
3 In vivo data suggested a possible acute activation of CYP3A4-catalyzed midazolam metabolism by efavirenz. efavirenz cytochrome P450 family 3 subfamily A member 4 Homo sapiens