Title : Effects of capsaicin and dihydrocapsaicin on human and rat liver microsomal CYP450 enzyme activities in vitro and in vivo.

Pub. Date : 2012

PMID : 22375877






2 Functional Relationships(s)
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1 In this study, we examined the inhibitory potentials of capsaicin and dihydrocapsaicin against CYP1A2, CYP2C9, CYP2C19, CYP2D6, CYP2E1, and CYP3A4/5 activities in human liver microsomes. Capsaicin cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 Time-dependent inhibition of CYP3A4/5 by capsaicin was found. Capsaicin cytochrome P450 family 3 subfamily A member 4 Homo sapiens