Title : Novel acrylonitrile derivatives, YHO-13177 and YHO-13351, reverse BCRP/ABCG2-mediated drug resistance in vitro and in vivo.

Pub. Date : 2011 Jul

PMID : 21566063






1 Functional Relationships(s)
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1 In contrast, it had no effect on P-glycoprotein-mediated paclitaxel resistance in MDR1-transduced human leukemia K562 cells and multidrug resistance-related protein 1-mediated doxorubicin resistance in MRP1-transfected human epidermoid cancer KB-3-1 cells. Doxorubicin ATP binding cassette subfamily C member 1 Homo sapiens