Title : Proposal of a new limited sampling strategy to predict CYP3A activity using a partial AUC of midazolam.

Pub. Date : 2010 Nov

PMID : 20680253






1 Functional Relationships(s)
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1 PURPOSE: Midazolam metabolic clearance to 1"-hydroxymidazolam is an accurate measure of CYP3A activity which requires extensive plasma and urine sampling. 1-hydroxymethylmidazolam cytochrome P450 family 3 subfamily A member 4 Homo sapiens