Title : Synthesis and in vivo evaluation of the putative breast cancer resistance protein inhibitor [11C]methyl 4-((4-(2-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl)phenyl)amino-carbonyl)-2-(quinoline-2-carbonylamino)benzoate.

Pub. Date : 2010 Jul

PMID : 20610168






1 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 Methyl is a recently discovered BCRP-selective inhibitor, which is structurally derived from the potent P-glycoprotein (P-gp) inhibitor tariquidar. tariquidar ATP binding cassette subfamily G member 2 (Junior blood group) Mus musculus