Title : Subtype-selective GABA(A) receptor modulation yields a novel pharmacological profile: the design and development of TPA023.

Pub. Date : 2009

PMID : 20230761






1 Functional Relationships(s)
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1 A drug-drug interaction study with itraconazole confirmed in vitro metabolic results implicating CYP3A enzymes as the major contributors to in vivo oxidative metabolism. Itraconazole cytochrome P450 family 3 subfamily A member 4 Homo sapiens