Title : Dose-response assessment of tariquidar and elacridar and regional quantification of P-glycoprotein inhibition at the rat blood-brain barrier using (R)-[(11)C]verapamil PET.

Pub. Date : 2010 May

PMID : 20016890






1 Functional Relationships(s)
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1 Regional differences in tariquidar-induced modulation of VPM brain uptake point to regional differences in cerebral P-gp function and expression in rat brain. tariquidar ATP-binding cassette, subfamily B (MDR/TAP), member 1B Rattus norvegicus