Title : Pre-clinical evaluation of cyclin-dependent kinase 2 and 1 inhibition in anti-estrogen-sensitive and resistant breast cancer cells.

Pub. Date : 2010 Jan 19

PMID : 20010939






1 Functional Relationships(s)
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1 Anti-estrogens, such as tamoxifen, antagonise estrogen-induced ERalpha transactivation of cyclin D1, resulting in reduced CDK4/6 activity, p27(Kip1)-mediated inhibition of CDK2 and growth arrest. Tamoxifen cyclin D1 Homo sapiens