Title : Synthesis, biological evaluation, X-ray structure, and pharmacokinetics of aminopyrimidine c-jun-N-terminal kinase (JNK) inhibitors.

Pub. Date : 2010 Jan 14

PMID : 19947601






1 Functional Relationships(s)
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1 The structure-activity relationships (SAR) around a series of aminopyrimidines were evaluated utilizing biochemical and cell-based assays to measure JNK inhibition and brain penetration in mice. 2-aminopyrimidine mitogen-activated protein kinase 8 Mus musculus