Title : Discovering potent small molecule inhibitors of cyclophilin A using de novo drug design approach.

Pub. Date : 2009 Sep 10

PMID : 19691347






1 Functional Relationships(s)
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1 The activities of the two most potent CypA inhibitors (3h and 3i) are 2.59 and 1.52 nM, respectively, which are about 16 and 27 times more potent than that of cyclosporin A. Tritium peptidylprolyl isomerase A Homo sapiens