Title : Synthesis, SAR study and biological evaluation of novel pyrazolo[1,5-a]pyrimidin-7-yl phenyl amides as anti-proliferative agents.

Pub. Date : 2009 Mar 1

PMID : 19200741






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1 We will present the synthesis, biological activities and SAR study of a series of pyrazolo[1,5-a]pyrimidines with an optimized phenyl amide moiety at the C-7 position. pyrazolo(1,5-a)pyrimidine sarcosine dehydrogenase Homo sapiens