Title : MTDL design strategy in the context of Alzheimer's disease: from lipocrine to memoquin and beyond.

Pub. Date : 2009

PMID : 19199985






2 Functional Relationships(s)
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1 Our first rationally designed MTDL was the polyamine caproctamine (1), which provided a synergistic cholinergic action against AD by antagonizing muscarinic M(2) autoreceptors and inhibiting acetylcholinesterase (AChE). Polyamines acetylcholinesterase (Cartwright blood group) Homo sapiens
2 Our first rationally designed MTDL was the polyamine caproctamine (1), which provided a synergistic cholinergic action against AD by antagonizing muscarinic M(2) autoreceptors and inhibiting acetylcholinesterase (AChE). Polyamines acetylcholinesterase (Cartwright blood group) Homo sapiens