Title : Cannabinoids desensitize capsaicin and mustard oil responses in sensory neurons via TRPA1 activation.

Pub. Date : 2008 Jan 30

PMID : 18234885






3 Functional Relationships(s)
Download
Sentence
Compound Name
Protein Name
Organism
1 Cannabinoids desensitize capsaicin and mustard oil responses in sensory neurons via TRPA1 activation. Capsaicin transient receptor potential cation channel, subfamily A, member 1 Mus musculus
2 The knockdown of TRPA1 activity in neurons completely eliminates the desensitizing effects of WIN and AM1241 on capsaicin-activated currents. Capsaicin transient receptor potential cation channel, subfamily A, member 1 Mus musculus
3 Furthermore, the WIN- or AM1241-induced inhibition of capsaicin-evoked nocifensive behavior via peripheral actions is reversed in TRPA1 null-mutant mice. Capsaicin transient receptor potential cation channel, subfamily A, member 1 Mus musculus