Title : Pharmacokinetic profile of temsirolimus with concomitant administration of cytochrome p450-inducing medications.

Pub. Date : 2007 Nov

PMID : 17913896






1 Functional Relationships(s)
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1 Because temsirolimus and its metabolite, sirolimus, are cytochrome P450 (CYP) 3A4/5 substrates, the potential exists for interaction with drugs that induce CYP3A activity, including enzyme inducers and rifampin. Sirolimus cytochrome P450 family 3 subfamily A member 4 Homo sapiens