Title : Sunitinib: a VEGF and PDGF receptor protein kinase and angiogenesis inhibitor.

Pub. Date : 2007 May 4

PMID : 17367763






2 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 Sunitinib (SU-11248, Sutent) inhibits at least eight receptor protein-tyrosine kinases including vascular endothelial growth factor receptors 1-3 (VEGFR1-VEGFR3), platelet-derived growth factor receptors (PDGFRalpha and PDGFRbeta), stem cell factor receptor (Kit), Flt-3, and colony-stimulating factor-1 receptor (CSF-1R). Sunitinib colony stimulating factor 1 receptor Homo sapiens
2 Sunitinib (SU-11248, Sutent) inhibits at least eight receptor protein-tyrosine kinases including vascular endothelial growth factor receptors 1-3 (VEGFR1-VEGFR3), platelet-derived growth factor receptors (PDGFRalpha and PDGFRbeta), stem cell factor receptor (Kit), Flt-3, and colony-stimulating factor-1 receptor (CSF-1R). Sunitinib colony stimulating factor 1 receptor Homo sapiens