Title : Poor correlation between 6beta-hydroxycortisol:cortisol molar ratios and midazolam clearance as measure of hepatic CYP3A activity.

Pub. Date : 2006 Aug

PMID : 16842393






2 Functional Relationships(s)
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1 AIMS: A non-invasive proposed method for measuring CYP3A activity is the urinary 6beta-hydroxycortisol:cortisol ratio. 6 beta-hydroxycortisol cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 Larger interindividual and intra-individual variability in CYP3A activity was observed in 6beta-hydroxycortisol:cortisol ratios compared with midazolam clearances. 6 beta-hydroxycortisol cytochrome P450 family 3 subfamily A member 4 Homo sapiens