Title : Discovery of 3,5-bis(trifluoromethyl)benzyl L-arylglycinamide based potent CCR2 antagonists.

Pub. Date : 2006 Jul 15

PMID : 16698264






2 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 Functionally, it blocked MCP-1 (CCL2)-induced calcium mobilization (IC50=50 nM) and chemotaxis mediated through the CCR2 receptor (9.6 nM). Calcium C-C motif chemokine ligand 2 Homo sapiens
2 Functionally, it blocked MCP-1 (CCL2)-induced calcium mobilization (IC50=50 nM) and chemotaxis mediated through the CCR2 receptor (9.6 nM). Calcium C-C motif chemokine ligand 2 Homo sapiens