Title : In vitro inhibitory effect of 1-aminobenzotriazole on drug oxidations catalyzed by human cytochrome P450 enzymes: a comparison with SKF-525A and ketoconazole.

Pub. Date : 2003

PMID : 15618748






1 Functional Relationships(s)
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1 In contrast, SKF-525A weakly inhibited CYP1A2-dependent activities (46% inhibition at 1200 microM) and CYP2E1-dependent activities (65% inhibition at 1000 microM). Proadifen cytochrome P450 family 1 subfamily A member 2 Homo sapiens