Title : Effect of St John's wort on imatinib mesylate pharmacokinetics.

Pub. Date : 2004 Oct

PMID : 15470331






1 Functional Relationships(s)
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1 Because imatinib is predominantly metabolized by cytochrome P450 (CYP) 3A4, its pharmacokinetics may be altered when it is coadministered with drugs or herbs (eg, St John"s wort) that modulate CYP3A4 activity. Imatinib Mesylate cytochrome P450 family 3 subfamily A member 4 Homo sapiens