Title : Impact of concentration and rate of intraluminal drug delivery on absorption and gut wall metabolism of verapamil in humans.

Pub. Date : 2004 Sep

PMID : 15371984






2 Functional Relationships(s)
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1 Moreover, intrinsic clearance of CYP3A4-mediated verapamil metabolism in homogenates of simultaneously collected shed enterocytes correlated with in vivo E GI of d0-verapamil 15 min /d3-verapamil 240 min (r = 0.62, P =.03). Verapamil cytochrome P450 family 3 subfamily A member 4 Homo sapiens
2 Moreover, intrinsic clearance of CYP3A4-mediated verapamil metabolism in homogenates of simultaneously collected shed enterocytes correlated with in vivo E GI of d0-verapamil 15 min /d3-verapamil 240 min (r = 0.62, P =.03). Verapamil cytochrome P450 family 3 subfamily A member 4 Homo sapiens