Title : Selective inhibition of CYP2B6-catalyzed bupropion hydroxylation in human liver microsomes in vitro.

Pub. Date : 2004 Jun

PMID : 15155554






1 Functional Relationships(s)
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1 In addition to CYP2B6, ticlopidine also inhibited both mephenytoin 4-hydroxylation (CYP2C19) (IC(50), 2.7 microM) and dextromethorphan O-demethylation (CYP2D6) (IC(50), 4.4 microM). Ticlopidine cytochrome P450 family 2 subfamily D member 6 Homo sapiens