Title : The allosteric potentiation of nicotinic acetylcholine receptors by galantamine is transduced into cellular responses in neurons: Ca2+ signals and neurotransmitter release.

Pub. Date : 2003 Nov

PMID : 14573772






1 Functional Relationships(s)
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1 Unlike galantamine, the acetylcholinesterase inhibitors rivastigmine and donepezil did not potentiate nAChR-mediated responses, whereas donepezil was a reasonably potent inhibitor of nicotine- and KCl-evoked increases in Ca2+. Rivastigmine acetylcholinesterase (Cartwright blood group) Homo sapiens