Title : Nonbenzamidine tetrazole derivatives as factor Xa inhibitors.

Pub. Date : 2003 Feb 10

PMID : 12565931






1 Functional Relationships(s)
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1 Herein we describe a series of tetrazole fXa inhibitors containing benzamidine mimics as the P(1) substrate, of which the aminobenzisoxazole moiety was found to be the most potent benzamidine mimic. 1H-tetrazole coagulation factor X Homo sapiens