Title : Inhibitors of vitamin D hydroxylases: structure-activity relationships.

Pub. Date : 2003 Feb 1

PMID : 12520539






1 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 Bulky substituents in alpha-position to the azole caused selectivity for CYP24, whereas bulky substituents in beta-position could result in selectivity for CYP27B. Azoles cytochrome P450 family 24 subfamily A member 1 Homo sapiens