Pub. Date : 2001 Oct
PMID : 11683901
4 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
1 | Chronic morphine exposure increases the phosphorylation of MAP kinases and the transcription factor CREB in dorsal root ganglion neurons: an in vitro and in vivo study. | Morphine | cAMP responsive element binding protein 1 | Rattus norvegicus |
2 | Naloxone effectively blocked these actions of morphine, whereas a selective MEK1 inhibitor, PD98059, inhibited the morphine-induced increase in the phosphorylation of ERK and CREB, and the expression of CGRP and SP. | Morphine | cAMP responsive element binding protein 1 | Rattus norvegicus |
3 | Naloxone effectively blocked these actions of morphine, whereas a selective MEK1 inhibitor, PD98059, inhibited the morphine-induced increase in the phosphorylation of ERK and CREB, and the expression of CGRP and SP. | Morphine | cAMP responsive element binding protein 1 | Rattus norvegicus |
4 | These in vitro and in vivo data suggest that the phosphorylation of MAP kinases and CREB plays a role in the morphine-induced increase in spinal CGRP and SP levels in primary sensory afferents, contributing to the development of tolerance to opioid-induced analgesia. | Morphine | cAMP responsive element binding protein 1 | Rattus norvegicus |