Pub. Date : 2001 Oct 11
PMID : 11585438
2 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
1 | Piperazine-based CCR5 antagonists as HIV-1 inhibitors. | Piperazine | C-C motif chemokine receptor 5 | Homo sapiens |
2 | Further optimization for pharmacokinetic properties afforded Sch-350634 (1), a prototypical piperazine-based CCR5 antagonist, which is a potent inhibitor of HIV-1 entry and replication in PBMCs. | Piperazine | C-C motif chemokine receptor 5 | Homo sapiens |