Title : Fluvoxamine is a potent inhibitor of tacrine metabolism in vivo.

Pub. Date : 1999 Jul

PMID : 10456487






3 Functional Relationships(s)
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Sentence
Compound Name
Protein Name
Organism
1 OBJECTIVE: In vitro studies have shown that tacrine is metabolized by cytochrome P4501A2 (CYP1A2). Tacrine cytochrome P450 family 1 subfamily A member 2 Homo sapiens
2 OBJECTIVE: In vitro studies have shown that tacrine is metabolized by cytochrome P4501A2 (CYP1A2). Tacrine cytochrome P450 family 1 subfamily A member 2 Homo sapiens
3 The aim of this study was to establish whether the potent CYP1A2 inhibitor fluvoxamine in clinically relevant doses could inhibit tacrine metabolism. Tacrine cytochrome P450 family 1 subfamily A member 2 Homo sapiens