Title : Enhancement of bradykinin and resensitization of its B2 receptor.

Pub. Date : 1999 Mar

PMID : 10082496






2 Functional Relationships(s)
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1 Administration of bradykinin or its ACE-resistant analogue desensitized the receptor, but it was resensitized (arachidonic acid release or [Ca2+]i mobilization) by agents such as enalaprilat (1 micromol/L). Arachidonic Acid kininogen 1 Homo sapiens
2 Enalaprilat resensitized the receptor via ACE to release arachidonic acid by bradykinin at a lower concentration (5 nmol/L) than required to mobilize [Ca2+]i (1 micromol/L). Arachidonic Acid kininogen 1 Homo sapiens